{"id":29727,"date":"2026-05-13T14:31:59","date_gmt":"2026-05-13T14:31:59","guid":{"rendered":"https:\/\/medicurahc.com\/product\/%e5%90%89%e7%91%9e%e6%9b%bf%e5%b0%bc-xospata%ef%bc%88everest%ef%bc%89\/"},"modified":"2026-05-13T14:31:59","modified_gmt":"2026-05-13T14:31:59","slug":"%e5%90%89%e7%91%9e%e6%9b%bf%e5%b0%bc-xospata%ef%bc%88everest%ef%bc%89","status":"publish","type":"product","link":"https:\/\/medicurahc.com\/zh-hans\/product\/%e5%90%89%e7%91%9e%e6%9b%bf%e5%b0%bc-xospata%ef%bc%88everest%ef%bc%89\/","title":{"rendered":"\u5409\u745e\u66ff\u5c3c\/Xospata\uff08Everest\uff09"},"content":{"rendered":"<h2>\ud83d\udc8a \u4ea7\u54c1\u6982\u89c8<\/h2>\n<p>\u5409\u7279\u66ff\u5c3c\uff08\u5546\u54c1\u540d\uff1aXospata\uff09\u662f\u4e00\u79cd\u53e3\u670d FMS \u6837\u916a\u6c28\u9178\u6fc0\u9176 3\uff08FLT3\uff09\u6291\u5236\u5242\uff0c\u4e3b\u8981\u7528\u4e8e\u6cbb\u7597\u643a\u5e26 FLT3 \u7a81\u53d8\u7684\u6210\u4eba\u6025\u6027\u9ad3\u7cfb\u767d\u8840\u75c5\uff08AML\uff09\u60a3\u8005\u3002<\/p>\n<p>Gilteritinib \u901a\u8fc7\u9009\u62e9\u6027\u6291\u5236\u7531 FLT3-ITD \u548c FLT3-TKD \u7a81\u53d8\u6fc0\u6d3b\u7684\u4fe1\u53f7\u901a\u8def\uff0c\u6709\u52a9\u4e8e\u6291\u5236\u767d\u8840\u75c5\u7ec6\u80de\u7684\u589e\u6b96\u4e0e\u5b58\u6d3b\u3002\u7531 Everest Pharma \u751f\u4ea7\u7684 Gilteritinib \u662f\u4e00\u6b3e\u9ad8\u8d28\u91cf\u4eff\u5236\u836f\uff0c\u5176\u6d3b\u6027\u6210\u5206\u76f8\u540c\u4e14\u7597\u6548\u76f8\u5f53\uff0c\u4e3a\u5168\u7403\u60a3\u8005\u63d0\u4f9b\u4e86\u4e00\u79cd\u66f4\u6613\u83b7\u53d6\u7684\u6cbb\u7597\u9009\u62e9\u3002 <\/p>\n<hr>\n<h2>\ud83c\udfaf \u4f5c\u7528\u673a\u5236\u4e0e\u4f18\u52bf<\/h2>\n<p>\u2705 \u540c\u65f6\u9776\u5411 FLT3-ITD \u548c FLT3-TKD \u7a81\u53d8<br \/>\n\u2705 \u540c\u65f6\u6291\u5236 AXL \u53d7\u4f53\u916a\u6c28\u9178\u6fc0\u9176\uff0c\u6709\u52a9\u4e8e\u964d\u4f4e\u6cbb\u7597\u8010\u836f\u6027\u3002<br \/>\n\u2705 \u53ef\u4f5c\u4e3a\u5355\u836f\u7597\u6cd5\u4f7f\u7528\uff0c\u4e5f\u53ef\u4f5c\u4e3a\u8054\u5408\u6cbb\u7597\u7b56\u7565\u7684\u4e00\u90e8\u5206\u3002<br \/>\n\u2705 \u591a\u9879\u4e34\u5e8a\u7814\u7a76\u5df2\u8bc1\u5b9e\u5e94\u7b54\u7387\u548c\u603b\u751f\u5b58\u671f\u5747\u6709\u6240\u6539\u5584\u3002<\/p>\n<p>Gilteritinib has been approved by the U.S. FDA and Japan PMDA and is included in NCCN guideline recommendations as a standard treatment option for relapsed or refractory FLT3-mutated AML.<\/p>\n<hr>\n<h2>\ud83d\udccc \u9002\u5e94\u75c7<\/h2>\n<p>\u5409\u745e\u66ff\u5c3c\u9002\u7528\u4e8e\uff1a<\/p>\n<ul>\n<li>\u7ecf\u7ecf\u9a8c\u8bc1\u7684\u5206\u5b50\u68c0\u6d4b\u786e\u8ba4\u4e3a\u643a\u5e26 FLT3 \u7a81\u53d8\uff08ITD \u6216 TKD\uff09\u7684\u590d\u53d1\u6027\u6216\u96be\u6cbb\u6027\u6025\u6027\u9ad3\u7cfb\u767d\u8840\u75c5\uff08AML\uff09\u6210\u4eba\u60a3\u8005<\/li>\n<\/ul>\n<p>\u5728\u5f00\u59cb\u6cbb\u7597\u524d\uff0c\u5e94\u4f7f\u7528\u7ecf\u8ba4\u8bc1\u7684\u5b9e\u9a8c\u5ba4\u68c0\u6d4b\u65b9\u6cd5\u786e\u8ba4 FLT3 \u7a81\u53d8\u72b6\u6001\u3002<\/p>\n<hr>\n<h2>\ud83d\udca1 \u5242\u91cf\u4e0e\u7ed9\u836f\u65b9\u6cd5<\/h2>\n<h3>\ud83d\udc65 1. \u60a3\u8005\u9009\u62e9 <\/h3>\n<ul>\n<li>\u6240\u6709\u60a3\u8005\u5728\u5f00\u59cb\u6cbb\u7597\u524d\u5747\u5e94\u63a5\u53d7 FLT3 \u7a81\u53d8\u68c0\u6d4b\u3002<\/li>\n<li>Therapy should be initiated under the supervision of a physician experienced in oncology treatment<\/li>\n<\/ul>\n<hr>\n<h3>\ud83d\udc8a 2. \u7ed9\u836f\u8bf4\u660e <\/h3>\n<ul>\n<li>\u53e3\u670d\u7247\u5242\u5242\u578b<\/li>\n<li>\u53ef\u968f\u9910\u6216\u7a7a\u8179\u670d\u7528<\/li>\n<li>\u8bf7\u6574\u7247\u541e\u670d\u836f\u7247\uff1b\u5207\u52ff\u63b0\u5f00\u3001\u538b\u788e\u6216\u5480\u56bc\u3002<\/li>\n<li>\u8bf7\u6bcf\u5929\u5728\u540c\u4e00\u65f6\u95f4\u670d\u7528\uff0c\u4ee5\u7ef4\u6301\u7a33\u5b9a\u7684\u836f\u7269\u6d53\u5ea6\u3002<\/li>\n<\/ul>\n<h3>\u6f0f\u670d\u836f\u7269\u6307\u5bfc<\/h3>\n<ul>\n<li>\u5982\u679c\u6f0f\u670d\uff0c\u8bf7\u5c3d\u5feb\u8865\u670d\uff0c\u5e76\u786e\u4fdd\u4e0e\u4e0b\u4e00\u6b21\u8ba1\u5212\u670d\u836f\u65f6\u95f4\u81f3\u5c11\u95f4\u9694 12 \u5c0f\u65f6\u3002<\/li>\n<li>\u5982\u679c\u670d\u836f\u540e\u53d1\u751f\u5455\u5410\uff0c\u8bf7\u52ff\u8ffd\u52a0\u5242\u91cf\uff1b\u6309\u8ba1\u5212\u7ee7\u7eed\u670d\u7528\u4e0b\u4e00\u6b21\u5242\u91cf\u3002<\/li>\n<li>\u5bf9\u4e8e\u9020\u8840\u5e72\u7ec6\u80de\u79fb\u690d\uff08HSCT\uff09\u540e\u6709\u590d\u53d1\u98ce\u9669\u7684\u60a3\u8005\uff0c\u5728\u9002\u5b9c\u60c5\u51b5\u4e0b\u53ef\u7ee7\u7eed\u6216\u91cd\u65b0\u5f00\u59cb\u5409\u7279\u66ff\u5c3c\uff08Gilteritinib\uff09\u6cbb\u7597\u3002<\/li>\n<\/ul>\n<hr>\n<h2>\ud83d\udcc8 \u5efa\u8bae\u5242\u91cf<\/h2>\n<table>\n<thead>\n<tr>\n<th>\u6cbb\u7597\u9636\u6bb5<\/th>\n<th>\u63a8\u8350\u5242\u91cf<\/th>\n<th>\u5907\u6ce8<\/th>\n<\/tr>\n<\/thead>\n<tbody>\n<tr>\n<td>\u521d\u59cb\u5242\u91cf<\/td>\n<td>120 mg\uff083 \u7247\uff09\uff0c\u6bcf\u65e5\u4e00\u6b21<\/td>\n<td>\u6bcf\u4e2a\u6cbb\u7597\u5468\u671f\u4e3a 28 \u5929<\/td>\n<\/tr>\n<tr>\n<td>\u5242\u91cf\u9012\u589e<\/td>\n<td>\u6700\u9ad8\u53ef\u8fbe 200 mg\uff085 \u7247\uff09\uff0c\u6bcf\u65e5\u4e00\u6b21<\/td>\n<td>\u82e5\u9996\u4e2a\u7597\u7a0b\u672a\u8fbe\u5230\u5b8c\u5168\u7f13\u89e3\uff0c\u53ef\u8003\u8651\u8fdb\u884c\u5242\u91cf\u9012\u589e<\/td>\n<\/tr>\n<\/tbody>\n<\/table>\n<p>\ud83d\udca1 \u901a\u5e38\u5efa\u8bae\u6301\u7eed\u6cbb\u7597\uff0c\u76f4\u81f3\u51fa\u73b0\u75be\u75c5\u8fdb\u5c55\u3001\u4e34\u5e8a\u83b7\u76ca\u4e27\u5931\u6216\u4e0d\u53ef\u8010\u53d7\u7684\u6bd2\u6027\u53cd\u5e94\u3002\u82e5\u672a\u83b7\u5f97\u65e9\u671f\u7f13\u89e3\uff0c\u53ef\u5728\u8bc4\u4f30\u7597\u6548\u524d\u8003\u8651\u8fdb\u884c\u6700\u591a 6 \u4e2a\u5468\u671f\u7684\u6cbb\u7597\u3002 <\/p>\n<hr>\n<h2>\ud83e\ude7a \u6cbb\u7597\u671f\u95f4\u7684\u76d1\u6d4b\u5efa\u8bae<\/h2>\n<h3>\u8840\u6db2\u68c0\u67e5\u4e0e\u751f\u5316\u76d1\u6d4b<\/h3>\n<ul>\n<li>\u5728\u5f00\u59cb\u6cbb\u7597\u4e4b\u524d<\/li>\n<li>\u5728\u7b2c\u4e00\u4e2a\u6cbb\u7597\u5468\u671f\u5185\u6bcf\u5468\u4e00\u6b21<\/li>\n<li>\u7b2c\u4e8c\u4e2a\u5468\u671f\u5185\u6bcf\u4e24\u5468\u4e00\u6b21<\/li>\n<li>\u5728\u968f\u540e\u7684\u6bcf\u4e2a\u5468\u671f\u4e4b\u524d<\/li>\n<\/ul>\n<h3>\u5fc3\u7535\u76d1\u6d4b<\/h3>\n<ul>\n<li>\u7b2c\u4e00\u4e2a\u5468\u671f\u7684\u7b2c8\u5929\u548c\u7b2c15\u5929<\/li>\n<li>\u5728\u968f\u540e\u7684\u6bcf\u4e2a\u5468\u671f\u4e4b\u524d<\/li>\n<\/ul>\n<p>\u82e5 QTcF \u95f4\u671f\u8d85\u8fc7 500 ms\uff0c\u5efa\u8bae\u4e2d\u65ad\u6cbb\u7597\u5e76\u8fdb\u884c\u4e34\u5e8a\u91cd\u65b0\u8bc4\u4f30\u3002<\/p>\n<hr>\n<h2>\u26a0\ufe0f \u91cd\u8981\u6ce8\u610f\u4e8b\u9879<\/h2>\n<ul>\n<li>Use caution when combined with medications known to prolong the QT interval<\/li>\n<li>\u5efa\u8bae\u5b9a\u671f\u76d1\u6d4b\u808c\u9178\u6fc0\u9176\u3001\u809d\u9176\u548c\u80be\u529f\u80fd\u3002<\/li>\n<li>\u598a\u5a20\u671f\u53ca\u54fa\u4e73\u671f\u7981\u7528\uff1b\u6cbb\u7597\u671f\u95f4\u5efa\u8bae\u91c7\u53d6\u6709\u6548\u7684\u907f\u5b55\u63aa\u65bd\u3002<\/li>\n<\/ul>\n<hr>\n<h2>\ud83d\udce6 \u5305\u88c5\u4e0e\u50a8\u5b58<\/h2>\n<ul>\n<li>Strength: 40 mg tablets<\/li>\n<li>\u5305\u88c5\uff1a\u6bcf\u74f6 90 \u7c92\uff08\u6309\u6bcf\u65e5 120 \u6beb\u514b\u7684\u5242\u91cf\u8ba1\u7b97\uff0c\u7ea6\u53ef\u670d\u7528 30 \u5929\uff09<\/li>\n<li>Storage: Store at room temperature away from moisture and direct light<\/li>\n<\/ul>\n<hr>\n<h2>\ud83d\udcda Additional Resources<\/h2>\n<p>\u6709\u5173\u6d89\u53ca\u5409\u7279\u66ff\u5c3c\uff08Gilteritinib\uff09\u7684\u4e34\u5e8a\u7597\u6548\u3001\u4e0d\u826f\u53cd\u5e94\u3001\u836f\u4ee3\u52a8\u529b\u5b66\u6216\u8054\u5408\u6cbb\u7597\u7814\u7a76\u7684\u66f4\u591a\u4fe1\u606f\uff0c\u8bf7\u53c2\u9605\uff1a<\/p>\n<ul>\n<li>NCCN \u6025\u6027\u9ad3\u7cfb\u767d\u8840\u75c5\u6307\u5357<\/li>\n<li><a href=\"https:\/\/clinicaltrials.gov\/?utm_source=chatgpt.com\">ClinicalTrials.gov <\/a>\u2014 \u6b63\u5728\u8fdb\u884c\u7684\u6025\u6027\u9ad3\u7cfb\u767d\u8840\u75c5\uff08AML\uff09\u4e34\u5e8a\u7814\u7a76\u53ca\u7814\u7a76\u8fdb\u5c55<\/li>\n<\/ul>\n","protected":false},"excerpt":{"rendered":"<p>\u5409\u745e\u66ff\u5c3c\uff08\u5546\u54c1\u540d\uff1aXospata\uff09\u662f\u4e00\u79cd\u53e3\u670d FMS \u6837\u916a\u6c28\u9178\u6fc0\u9176 3 (FLT3) \u6291\u5236\u5242\uff0c\u83b7\u6279\u7528\u4e8e\u6cbb\u7597\u4f34\u6709 FLT3 \u7a81\u53d8\u7684\u590d\u53d1\u6027\u6216\u96be\u6cbb\u6027\u6025\u6027\u9ad3\u7cfb\u767d\u8840\u75c5 (AML)\u3002<br \/>\n\u76ee\u524d\uff0c\u8be5\u836f\u7269\u6b63\u901a\u8fc7\u591a\u9879\u4e34\u5e8a\u8bd5\u9a8c\u79ef\u6781\u63a2\u7d22\u5176\u5728\u5176\u4ed6 AML \u4e9a\u578b\u53ca\u8054\u5408\u6cbb\u7597\u65b9\u6848\u4e2d\u7684\u5e94\u7528\uff0c\u5305\u62ec\u4e00\u7ebf\u6cbb\u7597\u3001\u7ef4\u6301\u6cbb\u7597\uff0c\u4ee5\u53ca\u4e0e\u5316\u7597\u6216\u5176\u4ed6\u9776\u5411\u7597\u6cd5\u8054\u5408\u4f7f\u7528\u3002<br \/>\nMedFind \u901a\u8fc7\u5408\u89c4\u7684\u56fd\u9645\u6e20\u9053\u63d0\u4f9b\u5409\u745e\u66ff\u5c3c\u7684\u6d77\u5916\u91c7\u8d2d\u670d\u52a1\uff0c\u5168\u7a0b\u6db5\u76d6\u5b8c\u6574\u7684\u7269\u6d41\u8ffd\u8e2a\u4e0e\u52a0\u5bc6\u9690\u79c1\u4fdd\u62a4\u3002<br \/>\n\u4e86\u89e3\u66f4\u591a\u5173\u4e8e\u9002\u5e94\u75c7\u3001\u4e34\u5e8a\u7597\u6548\u3001\u526f\u4f5c\u7528\u53ca\u7528\u836f\u6307\u5bfc\u7684\u4fe1\u606f\u3002<\/p>\n","protected":false},"featured_media":29728,"comment_status":"open","ping_status":"closed","template":"","meta":[],"product_brand":[],"product_cat":[110,135],"product_tag":[],"class_list":{"0":"post-29727","1":"product","2":"type-product","3":"status-publish","4":"has-post-thumbnail","6":"product_cat-110","7":"product_cat-135","9":"first","10":"instock","11":"sale","12":"shipping-taxable","13":"purchasable","14":"product-type-simple"},"_links":{"self":[{"href":"https:\/\/medicurahc.com\/zh-hans\/wp-json\/wp\/v2\/product\/29727","targetHints":{"allow":["GET"]}}],"collection":[{"href":"https:\/\/medicurahc.com\/zh-hans\/wp-json\/wp\/v2\/product"}],"about":[{"href":"https:\/\/medicurahc.com\/zh-hans\/wp-json\/wp\/v2\/types\/product"}],"replies":[{"embeddable":true,"href":"https:\/\/medicurahc.com\/zh-hans\/wp-json\/wp\/v2\/comments?post=29727"}],"version-history":[{"count":0,"href":"https:\/\/medicurahc.com\/zh-hans\/wp-json\/wp\/v2\/product\/29727\/revisions"}],"wp:featuredmedia":[{"embeddable":true,"href":"https:\/\/medicurahc.com\/zh-hans\/wp-json\/wp\/v2\/media\/29728"}],"wp:attachment":[{"href":"https:\/\/medicurahc.com\/zh-hans\/wp-json\/wp\/v2\/media?parent=29727"}],"wp:term":[{"taxonomy":"product_brand","embeddable":true,"href":"https:\/\/medicurahc.com\/zh-hans\/wp-json\/wp\/v2\/product_brand?post=29727"},{"taxonomy":"product_cat","embeddable":true,"href":"https:\/\/medicurahc.com\/zh-hans\/wp-json\/wp\/v2\/product_cat?post=29727"},{"taxonomy":"product_tag","embeddable":true,"href":"https:\/\/medicurahc.com\/zh-hans\/wp-json\/wp\/v2\/product_tag?post=29727"}],"curies":[{"name":"wp","href":"https:\/\/api.w.org\/{rel}","templated":true}]}}